Ligand efficiency
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Binding‐Site Purification of Actives (B‐SPA) Enables Efficient Large‐Scale Progression of Fragment Hits by Combining Multi‐Step Array Synthesis With HT Crystallography
Harold Grosjean, Anthony Aimon, Storm Hassell‐Hart, Warren Thompson, L. Koekemoer, James M. Bennett, A.R. Bradley, C.A. Anderson, Conor Wild, W.J. Bradshaw, Edward A. Fitzgerald, T. Krojer, O. Fedorov, Philip C. Biggin, John Spencer, F. von Delft
引用数: 9 • 2025