G protein-coupled receptor

Molecular Recognition of Corticotropin-releasing Factor by Its G-protein-coupled Receptor CRFR1

Augen A. Pioszak, Naomi R. Parker, Kelly Suino-Powell, H. Eric Xu

Citations: 150 • 2008

G protein-coupled receptor microarrays for drug discovery

Fang Ye, Joydeep Lahiri, Laurent Picard

Citations: 89 • 2003

Measuring Intracellular Calcium Fluxes in High Throughput Mode

Chris Chambers, Fiona Smith, Christine A. Williams, Sandra Marcos, Zhen Han Liu, Paul M. Hayter, Giuseppe Ciaramella, Wilma Keighley, Philip Gribbon, Andreas Sewing

Citations: 58 • 2003

Differential sensitivity of types 1 and 2 cholecystokinin receptors to membrane cholesterol

Ross M. Potter, Kaleeckal G. Harikumar, S. Vincent Wu, Laurence J. Miller

Citations: 57 • 2011

G-Protein-Coupled Receptor Microarrays

Fang Ye, Anthony G. Frutos, Joydeep Lahiri

Citations: 56 • 2002

Improving the apo-state detergent stability of NTS1 with CHESS for pharmacological and structural studies

Daniel J. Scott, Lutz Kummer, Pascal Egloff, Ross A. D. Bathgate, Andreas Plückthun

Citations: 39 • 2014

A 1,536-Well [ ³⁵ S]GTP <i>γ</i> S Scintillation Proximity Binding Assay for Ultra-High-Throughput Screening of an Orphan G <i>α</i> i-Coupled GPCR

Eric N. Johnson, Xiaoqing Shi, Jason Cassaday, Marc Ferrer, Berta Strulovici, Priya Kunapuli

Citations: 22 • 2008

Therapeutic Rescue of Misfolded/Mistrafficked Mutants

David C. Smithson, Jo Ann Janovick, P. Michael Conn

Citations: 19 • 2013

Screening a Plant Extract Library for Inhibitors of Cholecystokinin Receptor CCK1 Pathways

Alexandre Nesterov, Mei Hong, Carmen Hertel, Ping Jiao, Lidia Brownell, Edward Cannon

Citations: 15 • 2010

Membrane Biochips

Fang Ye, Anthony G. Frutos, Brian Webb, Yulong Hong, Ann M. Ferrie, Fang Lai, Joydeep Lahiri

Citations: 13 • 2002

High-throughput screening with a miniaturized radioligand competition assay identifies new modulators of human α2-adrenoceptors

Adyary Fallarero, Katariina Pohjanoksa, Gloria Wissel, Ulla-Mari Parkkisenniemi-Kinnunen, Henri Xhaard, Mika Scheinin, Pia Vuorela

Citations: 8 • 2012

Development of a Sensitive and HTS-Compatible Reporter Gene Assay for Functional Analysis of Human Adenosine A2a Receptors in CHO-K1 Cells

Yuting Tang, Jing-Qing Luo, Charles R. Fleming, Yan Kong, Gilbert C. Olini, Mary Jo Wildey, Druie Cavender, Keith T. Demarest

Citations: 8 • 2004

GPCR Assay Automation for Leveraging Lead Optimization

Mary Ellen Cvijic, Jing Chen, Steve Kubala, Joseph Nolfo, Garrett Kolodin, Litao Zhang

Citations: 5 • 2012